6-Fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-[4-methyl-2-(1-methylethyl)-3-pyridinyl]-4-[(2S)-2-methyl-4-(1-oxo-2-propen-1-yl)-1-piperazinyl]-pyrido[2,3-d]pyrimidin-2(1H)-one;
Sotorasib (AMG510) racemate is the racemate of AMG-510.
AMG-510 is a potent KRAS G12C covalent inhibitor with potential antitumor activity.