AMG 510

AMG 510

CAS No 2252403-56-6
Formula C30H30F2N6O3
Application

6-Fluoro-7-(2-fluoro-6-hydroxyphenyl)-1-[4-methyl-2-(1-methylethyl)-3-pyridinyl]-4-[(2S)-2-methyl-4-(1-oxo-2-propen-1-yl)-1-piperazinyl]-pyrido[2,3-d]pyrimidin-2(1H)-one;


Sotorasib (AMG510) racemate is the racemate of AMG-510.

AMG-510 is a potent KRAS G12C covalent inhibitor with potential antitumor activity.


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